(73) Merck Sharp & Dohme Corp., Rahway, NJ 07065-0907, 126 East Lincoln
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(72) WILSON, Kevin, Rahway NJ 07065-0907, 126 East Lincoln Avenue (US)
(72) DE ALMEIDA, Gabriela, Rahway NJ 07065-0907, 126 East Lincoln Avenue
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(72) HAIDLE, Andrew, Rahway NJ 07065-0907, 126 East Lincoln Avenue (US)
(72) KONRAD, Kaleen, Rahway NJ 07065-0907, 126 East Lincoln Avenue (US)
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(72) ZABIEREK, Anna, Rahway NJ 07065-0907, 126 East Lincoln Avenue (US)
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(73) IRM LLC, Hamilton HM 11, Hurst Holme 12 Trott Road (BM)
(54) DIE IMMUNREAKTION UNTERDRÜCKENDE VERBINDUNGEN UND
ZUSAMMENSETZUNGEN
(72) MI, Yuan, San diego, CA 92131, 11175 Affinity Court, Unit 45 (US)
(72) PAN, Shifeng, San Diego, CA 92130, 13880 Kerry Lane (US)
(72) GRAY, Nathanael, S., San Diego, CA 92122, 5652 Lamas Street (US)
(72) GAO, Wenqi, San Diego, CA 92123, 7958 Harmarsh Street (US)
(72) FAN, Yi, Poway, CA 92064, 12228 Pepper Tree Lane (US)
(72) JIANG, Tao, San Diego, CA 92130, 10721 Calle Mar De Mariposa (US)
(30) US 2003 05 19 471931 P
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(73) Takeda Pharmaceutical Company Limited, Osaka 541-0045, 1-1, Doshomachi
4-chome Chuo-ku Osaka-shi (JP)
(54) KONDENSIERTE RINGVERBINDUNGEN UND ANWENDUNG DAVON
(72) YASUMA, Tsuneo, Osaka-shi Osaka 532-8686, c/o TAKEDA
PHARMACEUTICAL COMPANY LIMITED 17-85, Jusohonmachi 2-chome
Yodogawa-ku (JP)
(72) TAKAKURA, Nobuyuki, Fujisawa Kanagawa 251-0012, c/o Takeda
Pharmaceutical Company Limited 26-1, Muraoka-Higashi 2-chome (JP)
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(73) Actelion Pharmaceuticals Ltd., 4123 Allschwil, Gewerbestrasse 16 (CH)
(54) THIAZOLDERIVATE UND IHRE VERWENDUNG ALS P2Y12 REZEPTOR
ANTAGONISTEN
(72) CAROFF, Eva, CH-4123 Allschwil, c/o Actelion Pharmaceuticals Ltd
Gewerbestrasse 16 (CH)
(72) HILPERT, Kurt, CH-4123 Allschwil, c/o Actelion Pharmaceuticals Ltd
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(72) HUBLER, Francis, CH-4123 Allschwil, c/o Actelion Pharmaceuticals Ltd
Gewerbestrasse 16 (CH)
(72) LEHMANN, David, CH-4123 Allschwil, c/o Actelion Pharmaceuticals Ltd
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(72) MEYER, Emmanuel, CH-4123 Allschwil, c/o Actelion Pharmaceuticals Ltd
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(72) RENNEBERG, Dorte, CH-4123 Allschwil, c/o Actelion Pharmaceuticals Ltd
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(73) F. Hoffmann-La Roche AG, 4070 Basel, Grenzacherstrasse 124 (CH)
(54) NEUE IMIDAZO[1,2-A]PYRIDIN- UND IMIDAZO[1,2-B]
PYRIDAZINDERIVATE
(72) DEWDNEY, Nolan, James, Saratoga California 95070, 14595 Horseshoe
Drive (US)
(72) LOU, Yan, San Jose California 95103, 1740 Fallbrook Avenue (US)
(72) SOTH, Michael, Milpitas California 95035, 2321 Edsel Drive (US)
(73) Piramal Enterprises Limited, Mumbai 400 013, Piramal Tower Ganpatrao
Kadam Marg Lower Parel (IN)
(54) Imidazo[4,5-c]chinolinderivate und ihre Verwendung bei der Behandlung von
Tumoren und/oder Entzündungen
(72) KUMAR, Sanjay, Mumbai 400063, Piramal Life Sciences Limited 1 Nirlon
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(72) VISHWAKARMA, Ram, Jammu 180001, Indian Institute of Integrative
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(72) MUNDADA, Ramswaroop, Mumbai 400063, Piramal Life Sciences Limited 1
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(72) DEORE, Vijaykumar, Mumbai 400063, Piramal Life Sciences Limited 1 Nirlon
Complex Off Western Express Highway Goregaon (East) (IN)
(72) KUMAR, Pramod, Mumbai 400063, Piramal Life Sciences Limited 1 Nirlon
Complex Off Western Express Highway Goregaon (East) (IN)
(72) SHARMA, Somesh, Mumbai 400063, Piramal Life Sciences Limited 1 Nirlon
Complex Off Western Express Highway Goregaon (East) (IN)
(73) Daiichi Sankyo Company, Limited, Toyko 103-8426, 3-5-1 Nihonbashi-honcho
Chuo-ku (JP)
(54) 3-(BIARYLOXY-)PROPIONSÄUREDERIVAT
(72) NISHI, Tatsuya, Shinagawa-ku Tokyo 140-8710, c/o DAIICHI SANKYO
COMPANY, LIMITED 1-2-58, Hiromachi (JP)
(72) NAKAMOTO, Yumi, Shinagawa-ku Tokyo 140-8710, c/o DAIICHI SANKYO
COMPANY, LIMITED 1-2-58, Hiromachi (JP)
(72) OCHIAI, Yuichi, Shinagawa-ku Tokyo 140-8710, c/o DAIICHI SANKYO
COMPANY, LIMITED 1-2-58, Hiromachi (JP)
(72) KITAZAWA, Ryoko, Shinagawa-ku Tokyo 140-8710, c/o DAIICHI SANKYO
COMPANY, LIMITED 1-2-58, Hiromachi (JP)
(72) HASEGAWA, Masashi, Edogawa-ku Tokyo 134-0081, c/o DAIICHI SANKYO
COMPANY, LIMITED 1-16-13, Kitakasai (JP)
(72) SUSAKI, Hiroshi, Edogawa-ku Tokyo 134-0081, c/o DAIICHI SANKYO RD
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(73) Abbvie Inc., North Chicago, IL 60064, 1 North Waukegan Road (US)
(54) PYRROLOPYRIDINE ALS INHIBITOREN VON KINASEN
(72) PENNING, Thomas D., Elmhurst Illinois 60126, 321 Highview (US)
(72) WOODS, Keith W., Libertyville Illinois 60048, 200 Red Top Drive Apt. 303
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(72) LAI, Chunqiu, Libertyville Illinois 60048, 1103 Tamarack Lane (US)
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(73) Sarepta Therapeutics, Inc., Bothell, Washington 98021, 3450 Monte Villa
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(54) VERFAHREN ZUR SYNTHESE VON MORPHOLINO-OLIGOMEREN
(72) FOX, Christina, Mary Josephine, Corvallis OR 97333, 30587 Stout Lane (US)
(72) REEVES, Matthew, Dale, Albany OR 97322, 2325 Edgemont Street SE (US)
(72) WELLER, Dwight, D., Corvallis OR 97330, 3323 N.W. Elmwood Drive (US)
(72) LI, Yongfu, Corvallis Oregon 97330, 2418 N.W. Estaview Circle (US)
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(73) IRM LLC, Hamilton, HM LX, 131 Front Street (BM)
(54) KONDENSIERTE IMIDAZOLE UND ZUSAMMENSETZUNGEN DIESE
ENTHALTEND ZUR BEHANDLUNG PARASITÄRER ERKRANKUNGEN, WIE Z.B.
MALARIA
(72) CHATTERJEE, Arnab K., San Diego California 92103, 1419 Essex Street, 2
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(72) NAGLE, Advait, San Diego California 92128, 12365 Springwater Point (US)
(72) WU, Tao, San Diego California 92122, 4162 Camino Ticino (US)
(72) TULLY, David, San Diego California 92130, 4278 Calle Isabelino (US)
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(73) LEO PHARMA A/S, 2750 Ballerup, Industriparken 55 (DK)
(54) NEUARTIGER PHOSPHODIESTERASE-HEMMER
(72) Felding, Jakob, DK-2920 Charlottenlund, Ordruphøjvej 24, 1 (DK)
(72) Nielsen, Simon, Feldbaek, DK-2730 Herlev, Afaldet 72 (DK)
(72) Larsen, Jens, Christian, Hojland, DK-2800 Lyngby, Sorgenfrigärdsvej 111C
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(72) Babu, Bollu, Ravindra, Andhra Pradesh, 31-Surya Enclave Thirumalagiri,
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(73) Pharma Mar S.A.U., 28770 Colmenar Viejo (Madrid), Avenida de los Reyes
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(54) Herstellung von natürlich vorkommenden Ecteinascidinen und verwandten
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(72) Menchaca, Roberto, E-28770, Madrid, Pharma Mar, S.A.U. Poligono Industrial
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(72) Martinez, Valentin, E-28770, Madrid, Pharma Mar, S.A.U. Poligono Industrial
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(72) Rodriguez, Alberto, E-28770, Madrid, Pharma Mar, S.A.U. Poligono Industrial
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(72) Rodriguez, Natividad, E-28770, Madrid, Pharma Mar, S.A.U. Poligono
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(72) Gallego, Pilar, E-28770, Madrid, Pharma Mar, S.A.U. Poligono Industrial La
Mina Avda. de los Reyes, 1 Colmenar Viejo (ES)
(72) Cuevas, Carmen, E-28770, Madrid, Pharma Mar, S.A.U. Poligono Industrial
La Mina Avda. de los Reyes, 1 Colmenar Viejo (ES)
(72) Munt, Simon, E-28770, Madrid, Pharma Mar, S.A.U. Poligono Industrial La
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(72) Manzanares, Ignacio, E-28770, Madrid, Pharma Mar, S.A.U. Poligono
Industrial La Mina Avda. de los Reyes 1 Colmenar Viejo (ES)
(30) GB 2002 02 04 0202544
Österreichisches Patentblatt 111. Jahrgang Nummer 4, Seite 1261
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