(73) Tokuyama Corporation, Shunan-shi, Yamaguchi-ken 745-8648, 1-1 Mikage-
cho (JP)
(54) VERBINDUNG MIT EINEM HYDANTOINRING UND
HERSTELLUNGSVERFAHREN DAFÜR
(72) SHIIGI, Hirofumi, Shunan-shi Yamaguchi 745-8648, c/o TOKUYAMA
CORPORATION 1-1 Mikage-cho (JP)
(72) SHIMAMURA, Mina, Shunan-shi Yamaguchi 745-8648, c/o TOKUYAMA
CORPORATION 1-1 Mikage-cho (JP)
(30) JP 2007 07 19 2007188157
(73) Akinion Pharmaceuticals AB, 171 77 Stockholm, Karolinska Institutet Science
Park (SE)
(54) PYRAZINE DERIVATE UND DEREN ANWENDUNG ALS PROTEIN KINASE
INHIBITOREN
(72) JENMALM JENSEN, Annika, S-756 45 Uppsala, Konsumvägen 37 B (SE)
(72) LEHMANN, Fredrik, S-193 33 Sigtuna, Stora Brännbovägen 48 (SE)
(72) NILSSON, Björn, M., S-112 49 Stockholm, Igeldammsgatan 20 (SE)
(72) NORDLING, Erik, S-182 35 Danderyd, Sportstugevägen 14A (SE)
(72) PARROW, Vendela, S-752 63 Uppsala, Ihres väg 9 (SE)
(30) SE 2008 02 01 0800250
(30) US 2008 04 04 123039 P
(30) SE 2008 05 21 0801185
(73) MediBeacon, LLC, St. Louis, MO 63108, 4041 Forest Park Avenue, Suite 250
(US)
(54) PYRAZINDERIVATE UND IHRE VERWENDUNG ZUR
NIERENÜBERWACHUNG
(72) NEUMANN, William, L., St. Louis, Missouri 63122, 212 W. Monroe (US)
(72) RAJAGOPALAN, Raghavan, St. Louis, Missouri 63146, 11432 A Tivoli Lane
(US)
(72) DORSHOW, Richard, B., St. Louis, Missouri 63146, 11977 Niehaus Lane
(US)
(30) US 2006 06 22 815712 P
(73) Merck Sharp & Dohme Corp., Rahway, NJ 07065-0907, 126 East Lincoln
Avenue (US)
(54) DIARYLTRIAZOLE ALS INHIBITOREN VON 11-BETA-HYDROXYSTEROID-
DEHYDROGENASE-1
(72) ASTER, Susan, D., Rahway, NJ 07065-0907, 126 East Lincoln Avenue (US)
(72) BALKOVEC, James, M., Rahway, NJ 07065-0907, 126 East Lincoln Avenue
(US)
(72) GRAHAM, Donald, W., Rahway, NJ 07065-0907, 126 East Lincoln Avenue
(US)
(72) GU, Xin, Rahway, NJ 07065-0907, 126 East Lincoln Avenue (US)
(72) KEVIN, Nancy, J., Rahway, NJ 07065-0907, 126 East Lincoln Avenue (US)
(72) PATEL, Gool, F., Rahway, NJ 07065-0907, 126 East Lincoln Avenue (US)
(72) PONPIPOM, Mitree, Rahway, NJ 07065-0907, 126 East Lincoln Avenue (US)
(30) US 2004 03 29 557344 P
(73) Merck Sharp & Dohme Corp., Rahway, NJ 07065-0907, 126 East Lincoln
Avenue (US)
(54) ALS INHIBITOREN VON FAAH GEEIGNETE OXAZOLDERIVATE
(72) CHOBANIAN, Harry, Rahway New Jersey 07065-0907, 126 East Lincoln
Avenue (US)
(72) LIN, Linus, S., Rahway New Jersey 07065-0907, 126 East Lincoln Avenue
(US)
(72) LIU, Ping, Rahway New Jersey 07065-0907, 126 East Lincoln Avenue (US)
(72) CHIODA, Marc, D., Rahway New Jersey 07065-0907, 126 East Lincoln
Avenue (US)
(72) DEVITA, Robert, J., Rahway New Jersey 07065-0907, 126 East Lincoln
Avenue (US)
(72) NARGUND, Ravi, P., Rahway New Jersey 07065-0907, 126 East Lincoln
Avenue (US)
(72) GUO, Yan, Rahway New Jersey 07065-0907, 126 East Lincoln Avenue (US)
(30) US 2008 08 04 137892 P
(73) Gilead Sciences, Inc., Foster City, CA 94404, 333 Lakeside Drive (US)
(54) 1'-SUBSTITUIERTE CARBA-NUKLEOSID-PRODRUGS ZUR ANTIVIRALEN
BEHANDLUNG
(72) CHO, Aesop, Mountain View CA 94040, 1656 Notre Dame Drive (US)
(72) KIM, Choung, U., San Carlos CA 94070, 1750 Elizabeth Street (US)
(72) RAY, Adrian, S., Redwood City CA 94065, 19 Pilot Circle (US)
(72) ZHANG, Lijun, Los Altos Hills CA 94022, 12525 Minorca Court (US)
(30) US 2011 05 26 201113117060
(30) US 2010 06 10 353351 P
(30) US 2010 05 28 349597 P
(30) US 2010 07 20 366041 P
(73) AbbVie Inc., North Chicago, IL 60064, 1 North Waukegan Road (US)
(54) Amid-Derivate als positive allosterische Modulatoren und
Verwendungsverfahren dafür
(72) Schrimpf, Michael, R., Grayslake, IL 60030, 327 Cambridge Drive (US)
(72) Mortell, Kathleen, H., Chicago, IL 60647, 2018 North Oakley Ave. (US)
(72) Nersesian, Diana, L., Gurnee, IL 60031, 4207 Coral Berry Path 103 (US)
(72) Lee, Chih-Hung, Vernon Hills, IL 60061, 569 South Central Park Place (US)
(72) Clapham, Bruce, Lindenhurst, IL 60046, 2813 Falling Waters Drive (US)
(30) US 2008 04 04 42323 P
(73) Eisai R&D Management Co., Ltd., Tokyo, 6-10, Koishikawa 4-chome Bunkyo-
ku (JP)
(54) ZWISCHENPRODUKTE UND VERFAHREN ZUR HERSTELLUNG VON
ZEARALENON-MAKROLID-ANALOGA
(72) BOIVIN, Roch, Lawrence MA 01843, 11 Oakland Road (US)
(72) CAMPAGNA, Silvio, A., Candia NH 03034, 621 Old Candia Road (US)
(72) DU, Hong, Andover MA 01810, 87 Chandler Road (US)
(72) FANG, Francis, G., Andover MA 01810, 16 Greybirch Road (US)
(72) HORSTMANN, Thomas, Boston MA 02116, 218 West Canton St. 4 (US)
(72) LEMELIN, Charles-Andre, North Chelmsford MA 01863, C-38 Scotty Hollow
Drive (US)
(72) LI, Jing, Andover MA 01810, 10b Washington Park Drive. (US)
(72) MCGUINNESS, Pamela, Methuen MA 01844, 8 Dracut Street (US)
(72) NIU, Xiang, MA 02148, 99 Florence Street Apt. 513 Malden (US)
(72) SCHNADERBECK, Matthew, J., Methuen MA 01844, 248 Lowell Street (US)
(72) WU, Kevin (kuo-ming), Acton MA 01820, 3 Kennedy Lane (US)
(72) ZHU, Xiaojie (jeff), Andover MA 01810, 12 Linda Road (US)
(30) US 2007 12 07 12408 P
(30) US 2007 12 07 12409 P
(30) US 2007 12 07 12411 P
(30) US 2008 07 11 80048 P
(73) Laboratorios Lesvi, S.L., 08970 Sant Joan Despí - Barcelona, Avda.
Barcelona 69 (ES)
(54) NEUARTIGES VERFAHREN ZUR HERSTELLUNG VON ASENAPIN
(72) DALMASES BARJOAN, Pere, E-08970 Sant Joan Despi, Av. Barcelona 69
(ES)
(72) HUGUET CLOTET, Juan, E-08970 Sant Joan Despi, Av. Barcelona 69 (ES)
(72) PEIRATS MASIA, Jordi, E-08970 Sant Joan Despi, Av. Barcelona 69 (ES)
(30) US 2010 08 04 370506 P
(30) EP 2010 07 29 10171222
(73) SCI Pharmatech, Inc., Taoyuan, Hai-Hu-Tsun Lu-Chu-Hsiang (TW)
(54) Verfahren zur Herstellung von (S)-(+)-N-Methyl-3-(1-naphthyloxy)-3-(2-
thienyl)-propylamin mittels einer optisch aktiven Methylhydroxylaminopropanol-
Verbindung als Zwischenprodukt
(72) Chen, Bo-Feng, Taoyuan, SCI Pharmtech, Inc. 186-2, Hai-Hu-Tsun Lu-Chu-
Hsiang (TW)
(72) Lu, Feng-Ju, Taoyuan, SCI Pharmtech, Inc. 186-2, Hai-Hu-Tsun Lu-Chu-
Hsiang (TW)
(72) Yeh, Jinun-Ban, Taoyuan, SCI Pharmatech, Inc. 186-2, Hai-Hu-Tsun Lu-Chu-
Hsiang (TW)
(72) Wong,, Weichyun, Toayuan, SCI Pharmtech, Inc. 186-2, Hai-Hu-Tsun Lu-
Chu-Hsiang (TW)
(73) Merck Sharp & Dohme Corp., Rahway, NJ 07065-0907, 126 East Lincoln
Avenue (US)
(54) SPIROPYRROLIDINDERIVATE ALS BETA-SEKRETASE-INHIBITOREN
ZUR BEHANDLUNG VON ALZHEIMER-KRANKHEIT
(72) LIU, Kun, New Jersey 07065-0907, Merck Sharp&Dohme Corp. 126 East
Lincoln Road Rahway (US)
(72) STACHEL, Shawn J., New Jersey 07065-0907, Merck Sharp&Dohme Corp.
126 EastLincoln Road Rahway (US)
(72) COBURN, Craig A., New Jersey 07065-0907, Merck Sharp&Dohme Corp. 126
East Lincoln Road Rahway (US)
(72) STEELE, Thomas G., New Jersey 07065-0907, Merck Sharp&Dohme Corp.
126 East Lincoln Road Rahway (US)
(72) SOLL, Richard, Shanghai 200131, 288 Fute Zhong Road Waigaoqiao Free
Trade Zone (CN)
(72) WU, Hao, Shanghai 200131, 288 Fute Zhong Road Waigaoqiao Free Trade
Zone (CN)
(72) PENG, Xuanjin, Shanghai 200131, 288 Fute Zhong Road Waigaoqiao Free
Trade Zone (CN)
(72) CAI, Yaxian, Shanghai 200131, 288 Fute Zhong Road Waigaoqiao Free Trade
Zone (CN)
(72) DU, Xiaoxing, Shanghai 200131, 288 Fute Zhong Road Waigaoqiao Free
Trade Zone (CN)
(72) LI, Jian, Shanghai 200131, 288 Fute Zhong Road Waigaoqiao Free Trade
Zone (CN)
(30) US 2009 02 20 208172
Österreichisches Patentblatt 111. Jahrgang Nummer 4, Seite 1020
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